10% Enrofloxacin
Kanema
Zochita za pharmacological
Enrofloxacin ndi battericidal wothandizira wa battericidal wa fluoroquinolone nyama. Kwa Esverherichia Coli, Salmonla, Klecellalla, Brucella, Actinoboccus a Accerus, Chruster, Zotsatira za pseudomonas Ainoginosa ndi streptococcus, komanso zofooka za mabakiteriya a Anaerobic. Zili ndi antibacteal mphamvu pa mabakiteriya omvera. Njira yoyeserera ya antibacterial ya mankhwalawa ndikuletsa bakiteriya kwa DNA ndikuphwanya ma bacteria a bacteri mosamala, polemba ndi kukonza ndikubwezera ndikubwezera. Mabakiteriya sangathe kukula ndikupanga nthawi zonse ndikufa.
Pharmacokinetics
10% Enrofloxacinimatha msanga komanso yolumikizidwa kwathunthu ndi jekeseni wa mu mnofu. Bioavailability wa malonda awa ndi 91.9% ya nkhumba ndi 82% ya ng'ombe zamkaka. Amagawidwa kwambiri mu nyama ndipo amatha kulowa ndi minofu. Kupatula kuchuluka kwa madzimadzi, mankhwalawa pafupifupi minofu yonse ndi apamwamba kuposa mu plasma. Chiphaso cha chiwindi chimayenera kuchotsa gulu la anthu 7yl la mphete 7 ya piprofloxacacin, kutsatiridwa ndi oxidation ndi glucuronic acid amamanga. Amakhala ndi impso (kudzera mwa aimpso kachulukidwe kachulukidwe), ndi 15% ~ 50% imachotsedwa mkodzo mu mawonekedwe ake oyamba. Kuthetsa theka la moyo kumasiyana kwambiri pakati pa nyama ndi njira zosiyanasiyana zoyang'anira. Kuthetsa theka-innicle jakisoni wa mnofu ndi ma 159 a ng'ombe, maola 9.9 mpaka 4,5 mpaka 4,5 maola a nkhosa, ndi maola 4.6 a nkhumba.
Kukhuzidwa
(1)10% Enrofloxacinimagwiritsidwa ntchito limodzi ndi aminoglycosides kapena penicillin, yomwe ili ndi matenda osokoneza bongo.
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Ntchito ndi kugwiritsa ntchito
Fluoroquinolone mankhwala. Amagwiritsidwa ntchito matenda a bakiteriya ndi minofu ya mycoplasma mu ziweto ndi nkhuku
Mlingo ndi makonzedwe
Jakisoni wa mnofu: Mlingo umodzi, pa 1 1,52Ml ng'ombe, nkhosa, ndi nkhumba; 0.025 ~ 0.05ml ya agalu, amphaka, ndi akalulu. Gwiritsani ntchito 1 mpaka 2 pa tsiku kwa masiku awiri mpaka atatu.
Zotsatira zoyipa
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(3) Zochita za khungu zimaphatikizapo Erythema, kuyabwa, urticaria ndi photossitativine.
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